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285 articles for Ambit Biosciences


The following articles (labelled with PubMed ID or TBD) are for your review
PMIDArticle TitlePublishedDeposition
21807507 4-Quinazolinyloxy-diaryl ureas as novel BRAFV600E inhibitors. 15-SEP-2011 29-AUG-2020
US9730937 RAF kinase modulator compounds and methods of use thereof 15-AUG-2017 23-JUN-2019
US9725465 Biaryl acetamide compounds and methods of use thereof 08-AUG-2017 12-JUN-2019
US9687494 Iminothiadiazine dioxide compounds as BACE inhibitors, compositions, and their use 27-JUN-2017 10-MAR-2018
US9295672 Optically active pyrazolylaminoquinazoline, and pharmaceutical compositions and methods of use thereof 29-MAR-2016 27-FEB-2017
US8551963 Imidazolothiazole compounds and methods of use thereof 08-OCT-2013 14-JAN-2014
22380736 Discovery of highly potent and selective pan-Aurora kinase inhibitors with enhanced in vivo antitumor therapeutic index. 12-APR-2012 17-MAY-2013
22168626 Identification of 1-(3-(6,7-dimethoxyquinazolin-4-yloxy)phenyl)-3-(5-(1,1,1-trifluoro-2-methylpropan-2-yl)isoxazol-3-yl)urea hydrochloride (CEP-32496), a highly potent and orally efficacious inhibitor of V-RAF murine sarcoma viral oncogene homologue B1 (BRAF) V600E. 09-FEB-2012 07-FEB-2013
18183025 A quantitative analysis of kinase inhibitor selectivity. 09-JAN-2008 25-DEC-2012
22037378 Comprehensive analysis of kinase inhibitor selectivity. 09-NOV-2011 19-JUL-2012
21802948 Novel series of pyrrolotriazine analogs as highly potent pan-Aurora kinase inhibitors. 22-AUG-2011 23-MAR-2012
19654408 AC220 is a uniquely potent and selective inhibitor of FLT3 for the treatment of acute myeloid leukemia (AML). 02-OCT-2009 11-JUN-2011
aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
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aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
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aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
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aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
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aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
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aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
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aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
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aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
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aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
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aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
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aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
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aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 23-APR-2011
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aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 21-APR-2011
aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 21-APR-2011
aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 21-APR-2011
aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 21-APR-2011
aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 21-APR-2011
aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 21-APR-2011
19646870 Arylcarboxyamino-substituted diaryl ureas as potent and selective FLT3 inhibitors. 17-AUG-2009 17-NOV-2010
19754199 Identification of N-(5-tert-butyl-isoxazol-3-yl)-N'-{4-[7-(2-morpholin-4-yl-ethoxy)imidazo[2,1-b][1,3]benzothiazol-2-yl]phenyl}urea dihydrochloride (AC220), a uniquely potent, selective, and efficacious FMS-like tyrosine kinase-3 (FLT3) inhibitor. 03-DEC-2009 30-AUG-2010
15711537 A small molecule-kinase interaction map for clinical kinase inhibitors. 14-MAR-2005 10-NOV-2009
aid1433 Kinase Inhibitor Selectivity Profiling Assay 21-NOV-2008 14-AUG-2009